1. Signaling Pathways
  2. GPCR/G Protein
  3. LPL Receptor
  4. LPAR5 Isoform
  5. LPAR5 Modulator

LPAR5 Modulator

LPAR5 Modulator (1):

Cat. No. Product Name Effect Purity
  • HY-W040176
    N-PTyrosine PA ammonium
    Modulator
    N-PTyrosine PA (N-Palmitoyl-tyrosine phosphoric acid) ammonium is a lysophosphatidic acid (LPA) receptor modulator, which exhibits weak inhibitory activity against LPA1 and partial agonist properties towards LPA5. N-PTyrosine PA ammonium inhibits the activation of LPA receptors and downstream responses by competing with agonists for binding sites. N-PTyrosine PA ammonium can induce morphological changes and aggregation, and also inhibit LPA-induced morphological changes through receptor desensitization caused by pre-incubation. N-PTyrosine PA ammonium can be used in the research of related diseases such as atherosclerosis and acute ischemic syndromes (e.g., unstable angina, myocardial infarction, stroke).